Terfenadine

CAS号

50679-08-8

分子式

C32H41NO2

主要靶点

Apoptosis|5-HT Receptor|Na+/Ca2+ Exchanger|HER|Histamine Receptor|Potassium Channel|Caspase|AChR

仅限科研使用

Cat No : CM00542

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Synonyms

PotassiumChannel|Potassium Channel|Na+ Exchanger|Na+/Ca2+ Exchanger|Na+Exchanger|MDL991|MDL-991|MDL 991|mAChR|Inhibitor|KcsA|Terfenadine|特非那定|Caspase|Ca2+Exchanger|Ca2+ Exchanger|Apoptosis|(±)-Terfenadine|5HTReceptor|5HT Receptor|HT|Histamine Receptor|HistamineReceptor|hERG|inhibit



产品信息

CAS号 50679-08-8
分子式 C32H41NO2
主要靶点 Apoptosis|5-HT Receptor|Na+/Ca2+ Exchanger|HER|Histamine Receptor|Potassium Channel|Caspase|AChR
主要通路 离子通道|凋亡|神经科学|G 蛋白偶联受体|神经科学|蛋白酶体|凋亡|JAK/STAT 信号通路|蛋白酪氨酸激酶|血管生成|离子通道|神经科学|免疫与炎症|G 蛋白偶联受体
分子量 471.67
纯度 99.75%, 此纯度可做参考,具体纯度与批次有关系,可咨询客服
储存条件 keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
别名 PotassiumChannel|Potassium Channel|Na+ Exchanger|Na+/Ca2+ Exchanger|Na+Exchanger|MDL991|MDL-991|MDL 991|mAChR|Inhibitor|KcsA|Terfenadine|特非那定|Caspase|Ca2+Exchanger|Ca2+ Exchanger|Apoptosis|(±)-Terfenadine|5HTReceptor|5HT Receptor|HT|Histamine Receptor|HistamineReceptor|hERG|inhibit

靶点活性

ERG (human):204 nM

溶解度

DMSO:47.2 mg/mL (100.07 mM)

参考文献

1.Kishimoto W, et al. Res Commun Mol Pathol Pharmacol. 1997 Dec;98(3):273-92.

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
=
×
×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
×
=
×
C1   V1   C2   V2