MEN 10207 acetate

CAS号

分子式

C59H72N14O12

主要靶点

Neurokinin receptor

仅限科研使用

Cat No : CM11553

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Synonyms

MEN10207 Acetate|MEN-10207 Acetate|MEN 10207 Acetate|MEN 10207 acetate|NK2|Neurokinin receptor|Neurokininreceptor



产品信息

CAS号
分子式 C59H72N14O12
主要靶点 Neurokinin receptor
主要通路 G 蛋白偶联受体|神经科学
分子量 1169.29
纯度 99.18%, 此纯度可做参考,具体纯度与批次有关系,可咨询客服
储存条件 keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
别名 MEN10207 Acetate|MEN-10207 Acetate|MEN 10207 Acetate|MEN 10207 acetate|NK2|Neurokinin receptor|Neurokininreceptor

体内活性

脊髓内注射神经激肽A和物质P以相似方式促进屈肌反射。对于脊髓内注射的神经激肽A(而非物质P),通过预先处理Men 10207醋酸盐[2]可以剂量依赖性地阻断反射的促进作用。

参考文献

1.Rovero P, Astolfi M, Renzetti AR, Patacchini R, Giachetti A, Maggi CA. Role of D-tryptophan for affinity of MEN 10207 tachykinin antagonist at NK2 receptors. Peptides. 1991 Sep-Oct;12(5):1015-8. doi: 10.1016/0196-9781(91)90053-r. PMID: 1666180.
2.Xu XJ, Maggi CA, Wiesenfeld-Hallin Z. On the role of NK-2 tachykinin receptors in the mediation of spinal reflex excitability in the rat. Neuroscience. 1991;44(2):483-90.

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