Talabostat mesylate

CAS号

150080-09-4

分子式

C10H23BN2O6S

主要靶点

Proteasome|DPP-4

仅限科研使用

Cat No : CM03796

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Synonyms

Dipeptidyl Peptidase|DPP|DPP4|DPP-4|inhibit|Talabostat|Talabostat Mesylate|Talabostat mesylate|Val-boroPro|Inhibitor|PT 100|PT100|PT-100



产品信息

CAS号 150080-09-4
分子式 C10H23BN2O6S
主要靶点 Proteasome|DPP-4
主要通路 蛋白酶体|泛素化|蛋白酶体
分子量 310.18
纯度 99.91%, 此纯度可做参考,具体纯度与批次有关系,可咨询客服
储存条件 Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
别名 Dipeptidyl Peptidase|DPP|DPP4|DPP-4|inhibit|Talabostat|Talabostat Mesylate|Talabostat mesylate|Val-boroPro|Inhibitor|PT 100|PT100|PT-100

靶点活性

DPP4:0.18 nM

溶解度

5% DMSO+95% Saline:2 mg/mL (6.45 mM);DMSO:60 mg/mL (193.44 mM)

参考文献

1.Cristillo AD, et al. HIV-1 Env vaccine comprised of electroporated DNA and protein co-administered with Talabostat. Biochem Biophys Res Commun. 2008 May 23;370(1):22-6.
2.Huang Y., et al. Fibroblast activation protein-α promotes tumor growth and invasion of breast cancer cells through non-enzymatic functions. Clin Exp Metastasis. 2011 Aug;28(6):567-79.
3.Meany H, et al. Pediatric phase I trial design using maximum target inhibition as the primary endpoint. J Natl Cancer Inst. 2010 Jun 16;102(12):909-12.

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
×
=
×
C1   V1   C2   V2