BRD4-IN-4

CAS号

304685-40-3

分子式

C17H18N2O3S

主要靶点

Epigenetic Reader Domain

仅限科研使用

Cat No : CM10891

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Synonyms

EpigeneticReaderDomain|Epigenetic Reader Domain|BRD4IN4|BRD4-IN-4|BRD4



产品信息

CAS号 304685-40-3
分子式 C17H18N2O3S
主要靶点 Epigenetic Reader Domain
主要通路 表观遗传
分子量 330.4
纯度 100%, 此纯度可做参考,具体纯度与批次有关系,可咨询客服
储存条件 Shipping with blue ice.
别名 EpigeneticReaderDomain|Epigenetic Reader Domain|BRD4IN4|BRD4-IN-4|BRD4

靶点活性

BRD4:6.83 μM

溶解度

DMSO:45 mg/mL (136.2 mM)

参考文献

1.Feng Y, et al. Design, synthesis and biological evaluation of benzo[cd]indol-2(1H)-ones derivatives as BRD4 inhibitors. Eur J Med Chem. 2018;152:264-273.

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
×
=
×
C1   V1   C2   V2