BRD4 Inhibitor-10

CAS号

1660117-38-3

分子式

C25H27N5O2

主要靶点

Epigenetic Reader Domain

仅限科研使用

Cat No : CM03962

Print datasheet

Synonyms

Inhibitor|BRD4 Inhibitor 10|BRD4 Inhibitor10|BRD-4 Inhibitor-10|BRD4 Inhibitor-10|BRD4-BD1|inhibit|Epigenetic Reader Domain|EpigeneticReaderDomain



产品信息

CAS号 1660117-38-3
分子式 C25H27N5O2
主要靶点 Epigenetic Reader Domain
主要通路 表观遗传
分子量 429.51
纯度 98.98%, 此纯度可做参考,具体纯度与批次有关系,可咨询客服
储存条件 Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
别名 Inhibitor|BRD4 Inhibitor 10|BRD4 Inhibitor10|BRD-4 Inhibitor-10|BRD4 Inhibitor-10|BRD4-BD1|inhibit|Epigenetic Reader Domain|EpigeneticReaderDomain

靶点活性

BRD4 BD1:8 nM

溶解度

DMSO:125 mg/mL (291.03 mM)

参考文献

1.Harald Engelhardt, et al. Pyridinones. WO2015022332A1.

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
=
×
×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
×
=
×
C1   V1   C2   V2